RATIONALLY DESIGNED 'DIPEPTOID' ANALOGUES OF CCK 'ALPHA'-METHYLTRYPTOPHAN DERIVATIVES AS HIGHLY SELECTIVE AND ORALLY ACTIVE GASTRIN AND CCK-B ANTAGONISTS WITH POTENT ANXIOLYTIC PROPERTIES
HORWELL, DAVID C.;HUGHES, JOHN;HUNTER, JOHN C.;PRITCHARD, MARTYN C.;RICHARDSON, REGINALD S.;ROBERTS, EDWARD;WOODRUFF, GEOFFREY N.
J. MED. CHEM., 34,(1991) N, C. 404-414
- DOI:
http://dx.doi.org/10.1021/jm00105a062